http://www.pharmachemm.com
Home > Products > Antipsychotic/Psychiatric/Mental > Tianeptine intermediate cas 66981-73-5 cas 1224690-84-9

Tianeptine intermediate cas 66981-73-5 cas 1224690-84-9

Product Description

Chemical Name: TIANEPTINE
Molecular Formula: C21H25ClN2O4S
Formula Weight: 436.95

CAS No.: 66981-73-5

66981-73-5



Chemical Name: tianeptine sulfate

Molecular Formula: 2(C21H25ClN2O4S).H2SO4.2(H2O)

Formula Weight:

CAS No.: 1224690-84-9

1224690-84-9



Tianeptine has antidepressant and anxiolytic effects with a relative lack of sedative, anticholinergic, and Cardiovascular side effects. It has been found to act as an atypical agonist of the μ-opioid receptor with clinically negligible effects on the δ- and κ-opioid receptors. μ-Opioid receptor agonists typically induce euphoria, and in accordance, tianeptine does so at high doses well above the normal therapeutic range.
Tianeptine is an antidepressant agent with a novel neurochemical profile. It increases serotonin (5-hydroxytryptamine; 5-HT) uptake in the brain (in contrast with most antidepressant agents) and reduces stress-induced atrophy of neuronal dendrites. Like the selective serotonin reuptake inhibitors (SSRIs) and in contrast with most tricyclic antidepressant agents, tianeptine does not appear to be associated with adverse cognitive, psychomotor, sleep, cardiovascular or bodyweight effects and has a low propensity for abuse. Tianeptine has a comparatively favourable pharmacokinetic profile. It is not subject to first-pass hepatic metabolism, has high bioavailability and limited distribution, and is rapidly eliminated. While this offers advantages for tianeptine over the tricyclic antidepressant agents in terms of dose titration, treatment changes and potential drug interactions, its rapid elimination makes adherence to dosage schedules more important.



Looking for ideal Tianeptineacid 99% EP Powder Manufacturer & supplier ? We have a wide selection at great prices to help you get creative. All the Coaxil Antidepressant Pharmceutical Intermediate are quality guaranteed. We are China Origin Factory of Tianeptine Hemisulfate Monohydrate. If you have any question, please feel free to contact us.

Product Categories : Antipsychotic/Psychiatric/Mental

Email to this supplier
  • *Subject:
  • *Messages:
    Your message must be between 20-8000 characters
Communicate with Supplier?Supplier
Mr. Vid Mr. Mr. Vid
What can I do for you?
Contact Supplier